SCHEMBL9302606

SCHEMBL9302606

CC(C)CN1C(=O)[C@@H](NC(=O)Oc2ccc([N+](=O)[O-])cc2)N=C(C2CCCCC2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 6/20 0.43
CCKBR P32239 11/20 0.42
OXTR P30559 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302596 1.00 BDKRB1 (0.43) BDKRB1CCKBROXTRALDH1A1LMNA
SCHEMBL9008655 1.00 BDKRB1 (0.43) BDKRB1CCKBROXTRALDH1A1LMNA
SCHEMBL9301875 1.00 BDKRB1 (0.43) BDKRB1CCKBROXTRALDH1A1LMNA
SCHEMBL9008654 1.00 BDKRB1 (0.43) BDKRB1CCKBROXTRALDH1A1LMNA
SCHEMBL9008657 1.00 BDKRB1 (0.43) BDKRB1CCKBROXTRALDH1A1LMNA
SCHEMBL9302408 0.90 BDKRB1 (0.45) BDKRB1CCKBROXTR
SCHEMBL9302403 0.90 BDKRB1 (0.45) BDKRB1CCKBROXTR
SCHEMBL9302412 0.90 BDKRB1 (0.45) BDKRB1CCKBROXTR
SCHEMBL8824652 0.90 BDKRB1 (0.54) BDKRB1CCKBR
SCHEMBL8824648 0.90 BDKRB1 (0.54) BDKRB1CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360802-A Antagonists of cholecystokinin and gastrin MERCK SHARPE & DOHME LTD. 1994-11-01 US disclosed
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP disclosed