SCHEMBL930705

SCHEMBL930705

COc1c(C)cc(C2(c3cccc(Cl)c3)NC(N)c3nccnc32)cc1C1CC1

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.32
HTR6 P50406 5/20 0.32
CHRNA1 P02708 2/20 0.30
CHRNG P07510 2/20 0.30
CHRNB1 P11230 2/20 0.30
CHRNB2 P17787 2/20 0.30
SLC6A2 P23975 2/20 0.30
CHRNB4 P30926 2/20 0.30
CHRNA3 P32297 2/20 0.30
CHRNA4 P43681 2/20 0.30
SLC6A3 Q01959 2/20 0.30
CHRND Q07001 2/20 0.30
SLC6A4 P31645 1/20 0.30
CTSD P07339 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931080 0.78
SCHEMBL930703 0.76 BACE1 (0.34) DPP4HTR6CTSDBACE1
SCHEMBL932098 0.74
SCHEMBL931363 0.74 BACE1 (0.52) CTSDBACE1
SCHEMBL929365 0.74 BACE1 (0.39) CTSDBACE1
SCHEMBL931144 0.74 BACE1 (0.39) CTSDBACE1
SCHEMBL931249 0.72 BACE1 (0.45) CTSDBACE1
SCHEMBL3358487 0.70 ALOX5AP (0.31) HTR6CTSDBACE1
SCHEMBL3356522 0.70
SCHEMBL3358408 0.69 OPRL1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed