SCHEMBL930784

SCHEMBL930784

CCOc1c(C)cc(C2(c3cccc(-c4cncnc4)c3)NC(N)c3nccnc32)cc1C

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.43
BACE2 Q9Y5Z0 5/20 0.43
SCN8A Q9UQD0 1/20 0.36
REN P00797 1/20 0.35
CTSD P07339 1/20 0.35
KCNH2 Q12809 5/20 0.35
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931363 0.91 BACE1 (0.52) BACE1BACE2SCN8ARENCTSD
SCHEMBL3359366 0.81 BACE1 (0.40) BACE1BACE2SCN8ARENCTSD
SCHEMBL929365 0.79 BACE1 (0.39) BACE1BACE2RENCTSDKCNH2
SCHEMBL931144 0.79 BACE1 (0.39) BACE1BACE2RENCTSDKCNH2
SCHEMBL3357766 0.78 BACE1 (0.41) BACE1BACE2KCNH2
SCHEMBL931347 0.78 BACE1 (0.52) BACE1BACE2KCNH2
SCHEMBL930938 0.78 BACE1 (0.52) BACE1BACE2KCNH2
SCHEMBL931387 0.78 BACE1 (0.52) BACE1BACE2KCNH2
SCHEMBL3357861 0.78 BACE1 (0.45) BACE1BACE2RENCTSDKCNH2
SCHEMBL931233 0.78 BACE1 (0.58) BACE1BACE2CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed