SCHEMBL9318232

SCHEMBL9318232

CCOC(=O)COc1ccc(CC(C)NCC(OC(=O)C(F)(F)F)c2cccc(Cl)c2)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 15/20 0.61
ADRB2 P07550 13/20 0.61
ADRB1 P08588 10/20 0.61
GLA P06280 1/20 0.61
CYP2D6 P10635 2/20 0.57
ADRA1D P25100 1/20 0.57
ADRA1A P35348 1/20 0.57
ADRA1B P35368 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
CYP3A4 P08684 1/20 0.56
HIF1A Q16665 1/20 0.56
SLC2A1 P11166 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9318460 0.92 ADRB3 (0.72) ADRB3ADRB2ADRB1GLACYP2D6
Trifluoroacetic Acid SCHEMBL9318231 0.87 ADRB3 (0.75) ADRB3ADRB2ADRB1GLACYP2D6
SCHEMBL9812024 0.85 ADRB3 (0.84) ADRB3ADRB2ADRB1GLACYP2D6
SCHEMBL9812022 0.85 ADRB3 (0.84) ADRB3ADRB2ADRB1GLACYP2D6
SCHEMBL9436811 0.85 ADRB3 (0.84) ADRB3ADRB2ADRB1GLACYP2D6
SCHEMBL10921498 0.82 ADRB3 (0.76) ADRB3ADRB2ADRB1GLACYP2D6
Hydrochloric Acid SCHEMBL10860449 0.81 ADRB3 (0.75) ADRB3ADRB2ADRB1GLACYP2D6
SCHEMBL10509636 0.81 ADRB3 (0.80) ADRB3ADRB2ADRB1GLACYP2D6
SCHEMBL10816420 0.81 ADRB3 (0.80) ADRB3ADRB2ADRB1GLACYP2D6
Hydrochloric Acid SCHEMBL10862129 0.80 ADRB3 (0.79) ADRB3ADRB2ADRB1GLACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347037-A (RR) and (RS stereoisomers of N-(7-ethoxycarbonylmethoxy-1,2,3,-tetrahydronaphth-2-yl)-2-(3-chlorophenyl)-2-hydroxyethanamine and their pharmaceutically acceptable salts SANOFI (FR) 1994-09-13 US disclosed
US-5041606-A Process for the O-alkylation of N-(hydroxy)aralkylphenylethanolamines SANOFI 1991-08-20 US disclosed
US-4927955-A Process for the O-alkylation of N-(hydroxy)aralkylphenylethanolamines SANOFI (FR) 1990-05-22 US disclosed