SCHEMBL9320893

SCHEMBL9320893

COC(=O)CC(=O)CC(O)/C=C/c1c(-c2ccc(F)cc2)c(COCc2ccccc2)c(=O)n(C)c1C(C)C

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.41
TBXA2R P21731 2/20 0.41
ADRA1A P35348 2/20 0.41
ESR1 P03372 1/20 0.41
CHRM1 P11229 1/20 0.41
PDE4A P27815 1/20 0.41
AR P10275 2/20 0.36
CYP2C9 P11712 3/20 0.35
SIRT6 Q8N6T7 2/20 0.35
ABCC3 O15438 1/20 0.35
ABCB11 O95342 1/20 0.35
PGR P06401 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
RXRA P19793 1/20 0.35
CCKAR P32238 1/20 0.35
PTGS2 P35354 1/20 0.35
NR4A2 P43354 1/20 0.35
PDE4D Q08499 1/20 0.35
SLC10A1 Q14973 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9665214 0.94 HMGCR (0.42) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL9665217 0.94 HMGCR (0.42) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL9318925 0.90 HMGCR (0.49) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL9662629 0.85 HMGCR (0.53) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL9662639 0.85 HMGCR (0.53) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL6956310 0.83 HMGCR (0.60) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL10650833 0.83 HMGCR (0.46) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL9318838 0.81 HMGCR (0.48) HMGCRTBXA2RADRA1AESR1CHRM1
SCHEMBL9321315 0.80 AR (0.43) AR
SCHEMBL9664046 0.80 AR (0.43) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0373423-B1 Substituted 2-pyridones and pyride-2-thiones, process for their preparation and their use in medicine BAYER AG (DE) 1994-01-12 EP disclosed
EP-0373423-A1 Substituted 2-pyridones and pyride-2-thiones, process for their preparation and their use in medicine BAYER AG (DE) 1990-06-20 EP disclosed