SCHEMBL9322784

SCHEMBL9322784

O=C1C2CCN(CC2)C1C(c1ccccc1)c1ccco1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 6/20 0.43
ALDH1A1 P00352 4/20 0.37
HPGD P15428 1/20 0.37
PKM P14618 1/20 0.37
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
RAB9A P51151 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14364967 0.85 MRGPRX1 (0.55) MRGPRX1ALDH1A1POLB
SCHEMBL2781629 0.85 MRGPRX1 (0.55) MRGPRX1ALDH1A1POLB
SCHEMBL6135225 0.85 MRGPRX1 (0.55) MRGPRX1ALDH1A1POLB
SCHEMBL9325051 0.78 MRGPRX1 (0.48) MRGPRX1ALDH1A1POLB
SCHEMBL9743327 0.77 MRGPRX1 (0.46) MRGPRX1
SCHEMBL5078507 0.77 MRGPRX1 (0.49) MRGPRX1
SCHEMBL8802582 0.76 MRGPRX1 (0.43) MRGPRX1
Benzylamine SCHEMBL28553128 0.76 MRGPRX1 (0.55) MRGPRX1
SCHEMBL9322829 0.76 MRGPRX1 (0.47) MRGPRX1ALDH1A1POLB
SCHEMBL700103 0.76 MRGPRX1 (0.46) MRGPRX1CHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0409931-B1 QUINUCLIDINE THERAPEUTIC AGENTS PFIZER (US) 1994-02-16 EP disclosed
US-5162339-A Substance P Antagonists, Gastrointestinal and Central Nervous System Disorders, Antiinflammatory Agents, Analgesics PFIZER INC. (US) 1992-11-10 US disclosed
WO-1990005525-A1 QUINUCLIDINE DERIVATIVES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1990-05-31 WO disclosed