SCHEMBL9325950

SCHEMBL9325950

Nc1nc(NCC2CC2)nc2nc(-c3ccco3)nn12

nearest known ligand 0.76

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.76
ADORA1 P30542 6/20 0.76
ADORA2B P29275 4/20 0.76
ADORA3 P0DMS8 4/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5421814 0.87 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5410869 0.85 ADORA2A (0.62) ADORA2AADORA1ADORA2BADORA3
SCHEMBL9325869 0.84 ADORA2A (0.76) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5418976 0.83 ADORA2A (0.58) ADORA2AADORA1ADORA2B
SCHEMBL9329035 0.83 ADORA2A (0.77) ADORA2AADORA1ADORA2BADORA3
SCHEMBL3544439 0.82
SCHEMBL9327307 0.82 ADORA2A (0.72) ADORA2AADORA1ADORA2BADORA3
SCHEMBL21936929 0.82 ADORA2A (0.74) ADORA2AADORA1ADORA2BADORA3
SCHEMBL7834626 0.82 ADORA2A (1.00) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5420803 0.81 ADORA2A (0.60) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed