SCHEMBL9327166

SCHEMBL9327166

CN(CCOc1ccc(C=C2SC(=O)NC2=O)cc1)c1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.80
HPGD P15428 7/20 0.67
PIM1 P11309 2/20 0.65
PIM2 Q9P1W9 2/20 0.65
PTPN1 P18031 2/20 0.62
POLB P06746 1/20 0.62
MAOA P21397 1/20 0.62
MAOB P27338 1/20 0.62
CISD1 Q9NZ45 2/20 0.60
AKR1B1 P15121 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9327162 1.00 PPARG (0.80) PPARGHPGDPIM1PIM2PTPN1
SCHEMBL9327176 0.88 PPARG (0.64) PPARGHPGDPIM1PIM2PTPN1
SCHEMBL1850981 0.87 PPARG (0.73) PPARGHPGDPIM1PIM2CISD1
SCHEMBL12520464 0.87 PPARG (0.73) PPARGHPGDPIM1PIM2CISD1
SCHEMBL1850984 0.87 PPARG (0.73) PPARGHPGDPIM1PIM2CISD1
SCHEMBL5111753 0.85 PPARG (0.78) PPARGHPGDPIM1PIM2CISD1
SCHEMBL1847035 0.85 PPARG (0.78) PPARGHPGDPIM1PIM2CISD1
SCHEMBL2260054 0.85 PPARG (0.78) PPARGHPGDPIM1PIM2CISD1
SCHEMBL6966749 0.85 HPGD (0.69) PPARGHPGDPIM1PIM2PTPN1
SCHEMBL6966747 0.85 HPGD (0.69) PPARGHPGDPIM1PIM2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415605-B1 Thiazolidinedione derivatives BEECHAM GROUP PLC (GB) 1994-03-02 EP disclosed
US-5132317-A Thiazolidinediones, Hypoglycemia Agents BEECHAM GROUP P.L.C. (GB) 1992-07-21 US disclosed
EP-0415605-A1 Thiazolidinedione derivatives Beecham Group p.l.c. (GB) 1991-03-06 EP disclosed