SCHEMBL9328835

SCHEMBL9328835

Cn1cnc2c1c(=O)[nH]c(=O)n2Cc1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.72
PDE4A P27815 1/20 0.66
ADORA2A P29274 1/20 0.66
PDE4B Q07343 1/20 0.66
PDE4C Q08493 1/20 0.66
PDE4D Q08499 1/20 0.66
KMT2A Q03164 5/20 0.65
MEN1 O00255 3/20 0.65
BRD2 P25440 1/20 0.58
BRD3 Q15059 1/20 0.58
BRDT Q58F21 1/20 0.58
MAPK1 P28482 2/20 0.57
CYP3A4 P08684 1/20 0.57
PMP22 Q01453 1/20 0.57
PNP P00491 1/20 0.56
KDM4E B2RXH2 4/20 0.55
POLB P06746 3/20 0.55
ADORA3 P0DMS8 2/20 0.54
BRAF P15056 1/20 0.54
ALDH1A1 P00352 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21389538 0.89 BRD4 (0.73) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL19090393 0.89 PDE4A (0.63) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL556233 0.84 BRD4 (0.82) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL19090444 0.84 BRD4 (1.00) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL12257284 0.81 PDE4A (0.80) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL6346663 0.81 ADORA2A (0.59) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL9351794 0.80 BRD4 (0.71) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL9351810 0.80 BRD4 (0.74) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL10571805 0.80 PDE4A (0.78) BRD4PDE4AADORA2APDE4BPDE4C
SCHEMBL7607643 0.79 PDE4A (0.74) BRD4PDE4AADORA2APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0319854-B1 Process for the methylation of xanthins BOEHRINGER INGELHEIM KG (DE) 1994-03-02 EP disclosed
EP-0319854-A2 Process for the methylation of xanthins BOEHRINGER INGELHEIM KG (DE) 1989-06-14 EP disclosed