Coumarin

Coumarin

SCHEMBL9330710

Cc1c(-c2ccccc2)c(=O)oc2ccccc12.O=c1ccc2ccccc2o1

nearest known ligand 0.54

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERAP1 Q9NZ08 1/20 0.54
TDP1 Q9NUW8 2/20 0.54
CA1 P00915 2/20 0.54
CA2 P00918 2/20 0.54
CA12 O43570 1/20 0.54
LMNA P02545 1/20 0.54
CA3 P07451 1/20 0.54
CA4 P22748 1/20 0.54
CA6 P23280 1/20 0.54
CA5A P35218 1/20 0.54
CA7 P43166 1/20 0.54
MCL1 Q07820 1/20 0.54
CA9 Q16790 1/20 0.54
SOST Q9BQB4 1/20 0.54
CA14 Q9ULX7 1/20 0.54
CA5B Q9Y2D0 1/20 0.54
KDM4E B2RXH2 6/20 0.46
ALDH1A1 P00352 4/20 0.46
PGR P06401 4/20 0.46
KMT2A Q03164 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4449250 0.87 ERAP1 (0.68) ERAP1CA1CA2CA12LMNA
Coumarin SCHEMBL2121277 0.80 CA1 (0.65) TDP1CA1CA2CA12LMNA
SCHEMBL7912329 0.76 HPGD (0.57) ERAP1LMNAKDM4EALDH1A1KMT2A
SCHEMBL7121658 0.76 CA1 (0.56) ERAP1CA1CA2CA9KDM4E
SCHEMBL7358531 0.75 CA12 (0.95) ERAP1TDP1CA1CA2CA12
Coumarin SCHEMBL19183240 0.75 CA12 (0.95) ERAP1TDP1CA1CA2CA12
SCHEMBL19484976 0.75 CYP1B1 (0.60) ERAP1CA1CA2CA12CA9
Coumarin SCHEMBL28286390 0.74 CA12 (0.77) ERAP1TDP1CA1CA2CA12
Coumarin SCHEMBL29182492 0.74 CA12 (0.91) ERAP1TDP1CA1CA2CA12
Coumarin SCHEMBL25431834 0.74 CA12 (0.91) ERAP1TDP1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0592583-A1 METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1994-04-20 EP disclosed
WO-1993000896-A1 METHOD FOR THE INHIBITION OF ALDH-I USEFUL IN THE TREATMENT OF ALCOHOL DEPENDENCE OR ALCOHOL ABUSE THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1993-01-21 WO disclosed