SCHEMBL9339010

SCHEMBL9339010

Fc1ccc2sc(COc3cccc(CBr)c3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.56
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KMT2A Q03164 1/20 0.53
CYSLTR1 Q9Y271 7/20 0.49
CYSLTR2 Q9NS75 6/20 0.49
L3MBTL1 Q9Y468 2/20 0.48
MAPK1 P28482 1/20 0.48
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
GRM5 P41594 1/20 0.41
MAOB P27338 1/20 0.41
ALOX5 P09917 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339227 0.88 PTGER4 (0.58) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9339029 0.87 PTGER4 (0.55) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9334986 0.83 PTGER4 (0.54) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9335208 0.83 NPC1 (0.55) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9754811 0.83 NPC1 (0.55) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
Bromide SCHEMBL9339050 0.82 PTGER4 (0.52) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9335068 0.79 SMN1; SMN2 (0.53) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9334993 0.78 PTGER4 (0.53) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9336045 0.78 PTGER4 (0.55) PTGER4NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL9339025 0.78 PTGER4 (0.53) PTGER4NPC1RAB9ASMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533695-B1 IMIDAZO (4,5-c) PYRIDINES WITH PAF ANTAGONIST ACTIVITY PFIZER (US) 1994-10-05 EP disclosed
US-5322847-A Inhibit platelet activating factor, block leukotriene D4 receptors PFIZER INC. (US) 1994-06-21 US disclosed
EP-0533695-A1 IMIDAZO (4,5-c) PYRIDINES WITH PAF ANTAGONIST ACTIVITY. PFIZER (US) 1993-03-31 EP disclosed
WO-1991017163-A1 IMIDAZO (4,5-c) PYRIDINES WITH PAF ANTAGONIST ACTIVITY PFIZER INC. (US) 1991-11-14 WO disclosed