SCHEMBL9339019

SCHEMBL9339019

CCCCCCc1nc2cc(CCCCC)c(=O)c(CCCCC)cc2n1Cc1ccc(-c2ccccc2C(=O)O)cc1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 7/20 0.75
AGTR1 P30556 2/20 0.69
AGTR2 P50052 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9335510 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9337424 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9335221 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9335223 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9335193 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9335587 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9339075 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9335483 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9335583 1.00 PPARG (0.75) PPARGAGTR1AGTR2
SCHEMBL9339351 1.00 PPARG (0.75) PPARGAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432737-A1 Cycloheptimidazolone compounds as angiotensin II antagonists for control of hypertension G.D. Searle & Co. (US) 1991-06-19 EP claimed
US-5281615-A Hypotensive agents G. D. SEARLE & CO. (US) 1994-01-25 US disclosed
US-5104891-A CYCLOHEPTIMIDAZOLONE COMPOUNDS AS ANGIOTENSIN II ANTAGONISTS FOR CONTROL OF HYPERTENSION G. D. SEARLE & CO. (US) 1992-04-14 US disclosed