SCHEMBL9339241

SCHEMBL9339241

[NH]Cc1ccc2c(c1)OCCCO2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
KDM1A O60341 1/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
CYP2D6 P10635 2/20 0.44
TAAR1 Q96RJ0 3/20 0.43
ALDH1A1 P00352 4/20 0.42
GAA P10253 2/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
HPGD P15428 2/20 0.42
CASP3 P42574 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SLC6A4 P31645 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4181991 0.92 CYP2D6 (0.50) CYP1A2CYP3A4MAPTKDM1AMAOA
SCHEMBL2774556 0.83 CYP3A4 (0.63) CYP1A2CYP3A4MAPTCYP2D6TAAR1
SCHEMBL9335512 0.82 TAAR1 (0.46) CYP1A2CYP3A4MAPTKDM1AMAOA
SCHEMBL3820698 0.80 CYP1A2 (0.46) CYP1A2CYP3A4MAPTKDM1AMAOA
SCHEMBL1174021 0.80 CYP2D6 (0.47) CYP1A2CYP3A4MAPTKDM1AMAOA
SCHEMBL111534 0.80 TAAR1 (0.52) CYP1A2CYP3A4MAPTKDM1AMAOA
SCHEMBL8918332 0.80 NPC1 (0.47) MAPTKDM1AMAOAMAOBCYP2D6
SCHEMBL30896292 0.80 KDM1A (0.46) CYP1A2CYP3A4MAPTKDM1AMAOA
SCHEMBL3083264 0.80 PDCD1 (0.50) CYP3A4KDM1AMAOAMAOBCYP2D6
SCHEMBL3023636 0.77 TAAR1 (0.49) CYP1A2CYP3A4MAPTKDM1AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0394440-B1 PHENYLCARBOXYLIC ACID DERIVATIVES OTSUKA PHARMA CO LTD (JP) 1994-05-11 EP disclosed
US-4999378-A Antilipemic, anticholesterol, antidiabetic, treatment of atherosclerosis and obesity OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1991-03-12 US disclosed