SCHEMBL936412

SCHEMBL936412

CN1CCN(c2ccc(-c3cc(-c4cccc5c4CCNC5=O)n[nH]3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.59
PRKD1 Q15139 9/20 0.53
MAP4K1 Q92918 1/20 0.46
MAPK1 P28482 1/20 0.43
MAP2K1 Q02750 1/20 0.43
PARP1 P09874 2/20 0.43
PARP10 Q53GL7 2/20 0.43
PARP11 Q9NR21 2/20 0.43
FLT3 P36888 4/20 0.42
AURKA O14965 3/20 0.42
KDR P35968 3/20 0.42
JAK2 O60674 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19951651 0.74 MELK (0.79) MELKPRKD1MAP4K1FLT3AURKA
SCHEMBL28977159 0.74 MELK (0.82) MELKPRKD1MAP4K1MAPK1FLT3
SCHEMBL28977172 0.74 MELK (0.86) MELKPRKD1MAP4K1FLT3AURKA
SCHEMBL28977186 0.73 MELK (0.77) MELKPRKD1MAP4K1JAK2
SCHEMBL30775205 0.73 KDR (0.49) MELKPARP1FLT3AURKAKDR
SCHEMBL998233 0.72 PRKD1 (0.74) MELKPRKD1MAP4K1FLT3AURKA
SCHEMBL1081001 0.72 PRKD1 (0.73) MELKPRKD1MAP4K1FLT3AURKA
SCHEMBL27741315 0.71 MELK (0.73) MELKPRKD1MAP4K1
SCHEMBL28977183 0.71 MELK (0.76) MELKPRKD1MAP4K1FLT3AURKA
SCHEMBL28977178 0.71 MELK (0.72) MELKPRKD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009484-A1 ARYLPYRAZOLES AND ARYLISOXAZOLES AND THEIR USE AS PKD MODULATORS NOVARTIS AG (CH) 2011-01-27 WO disclosed