SCHEMBL9364670

SCHEMBL9364670

NS(=O)(=O)c1cc2c(cc1C(F)(F)F)[nH]c(=O)c(=O)n2O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.43
CA9 Q16790 3/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
GRIA1 P42261 6/20 0.39
GRIA2 P42262 6/20 0.39
GRIA3 P42263 6/20 0.39
GRIA4 P48058 6/20 0.39
GRIK1 P39086 3/20 0.39
GRIK2 Q13002 3/20 0.39
GRIK3 Q13003 3/20 0.39
GRIK5 Q16478 3/20 0.39
GRIK4 Q16099 2/20 0.39
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9364672 0.78 GRIA1 (0.45) CA12CA9GRIA1GRIA2GRIA3
SCHEMBL9365197 0.77 GRIA1 (0.40) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL9091900 0.75 GRIA1 (0.40) CA12CA9GRIA1GRIA2GRIA3
SCHEMBL9365202 0.74 GRIA1 (0.40) GRIA1GRIA2GRIA3GRIA4GRIK1
SCHEMBL9370056 0.71 PARG (0.45) CA12CA9CA1CA2ALDH1A1
SCHEMBL6927437 0.69 CA1 (0.41) CA12CA9CA1CA2CA4
SCHEMBL9826888 0.69 CA12 (0.56) CA12CA9ALDH1A1CYP2C9SMN1; SMN2
SCHEMBL9080167 0.69 CA12 (0.52) CA12CA9KDM4EALDH1A1CYP2C9
SCHEMBL6927443 0.67 CA12 (0.41) CA12CA9CA1CA2CA4
SCHEMBL9362821 0.67 KDM4E (0.31) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377112-B1 Quinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-08-24 EP claimed
US-5061706-A 2,3-QUINOXALINEDIONES FOR USE AS NEUROLEPTICS NOVO NORDISK A/S (DK) 1991-10-29 US claimed
US-20250288544-A1 PROBENECID FOR USE IN TREATING EPILEPTIC DISEASES, DISORDERS OR CONDITIONS PARIS SCIENCES ET LETTRES - QUARTIER LATIN (FR) 2025-09-18 US disclosed
US-12318358-B2 Probenecid for use in treating epileptic diseases, disorders or conditions PARIS SCIENCES ET LETTRES (FR) 2025-06-03 US disclosed
CN-111386107-A Use of probenecid in the treatment of an epileptic disease, disorder or condition 巴黎科技与文学─拉丁区 2020-07-07 CN disclosed
US-20200163916-A1 PROBENECID FOR USE IN TREATING EPILEPTIC DISEASES, DISORDERS OR CONDITIONS PARIS SCIENCES ET LETTRES - QUARTIER LATIN (FR) 2020-05-28 US disclosed
EP-0377112-B1 Quinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-08-24 EP disclosed
US-5061706-A 2,3-QUINOXALINEDIONES FOR USE AS NEUROLEPTICS NOVO NORDISK A/S (DK) 1991-10-29 US disclosed
EP-0377112-A1 Quinoxaline compounds and their preparation and use NOVO NORDISK A/S (DK) 1990-07-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200163916-A1 PROBENECID FOR USE IN TREATING EPILEPTIC DISEASES, DISORDERS OR CONDITIONS NLN, CLN6, SLC1A2 CA12 285/4885CA9 702/4885CA1 97/4885
US-20250288544-A1 PROBENECID FOR USE IN TREATING EPILEPTIC DISEASES, DISORDERS OR CONDITIONS NLN, CLN6, SLC1A2 CA12 285/4885CA9 702/4885CA1 97/4885
US-12318358-B2 Probenecid for use in treating epileptic diseases, disorders or conditions NLN, CLN6, SLC1A2 CA12 285/4885CA9 702/4885CA1 97/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.