SCHEMBL9366605

SCHEMBL9366605

C=C[C@H]1CO[C@H](c2ccc(-c3ccc(F)c(F)c3)nc2)OC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 13/20 0.42
GRM2 Q14416 1/20 0.38
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
MAOB P27338 5/20 0.33
NSD2 O96028 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9366617 1.00 KDM1A (0.42) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9366249 0.86 GRIA2 (0.38) KDM1ACYP11B1CYP11B2NPC1MAOB
SCHEMBL9366242 0.86 GRIA2 (0.38) KDM1ACYP11B1CYP11B2NPC1MAOB
SCHEMBL9732702 0.86 KDM1A (0.41) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9366647 0.86 KDM1A (0.41) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9366637 0.86 KDM1A (0.41) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9732698 0.86 KDM1A (0.41) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9365271 0.85 KDM1A (0.38) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9365278 0.85 KDM1A (0.38) KDM1AGRM2CYP11B1CYP11B2KDM4E
SCHEMBL9365229 0.84 KDM1A (0.50) KDM1AKDM4ENPC1RAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433835-B1 Dioxanylpyridines HOFFMANN LA ROCHE (CH) 1994-05-18 EP disclosed
US-5160661-A DIOXANYLPYRIDINE HOFFMANN-LA ROCHE INC. (US) 1992-11-03 US disclosed
EP-0433835-A2 Dioxanylpyridines F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed