SCHEMBL9378221

SCHEMBL9378221

NC(=O)OC1c2ccccc2CCC1I

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.42
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
PIN1 Q13526 3/20 0.39
HSD11B1 P28845 2/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
RET P07949 1/20 0.38
HTR2A P28223 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378215 1.00 IDO1 (0.42) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL19911672 0.83 IDO1 (0.44) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL19911693 0.83 IDO1 (0.47) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL19911668 0.83 IDO1 (0.44) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL19911692 0.83 IDO1 (0.47) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL9373549 0.83 IDO1 (0.44) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL9373544 0.83 IDO1 (0.44) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL2175357 0.78 IDO1 (0.61) IDO1PIN1HSD11B1CA1CA2
SCHEMBL19911670 0.74 IDO1 (0.47) IDO1CHRM2CHRM1CHRM3PIN1
SCHEMBL19911671 0.74 IDO1 (0.47) IDO1CHRM2CHRM1CHRM3PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0546123-A4 1994-04-27 EP disclosed
EP-0546123-A1 ALPHA-SUBSTITUTED TRYPTOPHANE DIPEPTOID DERIVATIVES WARNER-LAMBERT COMPANY (US) 1993-06-16 EP disclosed
WO-1992004322-A1 ALPHA-SUBSTITUTED TRYPTOPHANE DIPEPTOID DERIVATIVES WARNER-LAMBERT COMPANY (US) 1992-03-19 WO disclosed