SCHEMBL938071

SCHEMBL938071

CC1CCC(C(=O)N(c2cc(C#CC(C)(C)C)sc2C(=O)O)C2CCC(Oc3cc(CN4CCC(O)C4)ccn3)CC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.51
CYP2E1 P05181 1/20 0.46
MLNR O43193 5/20 0.32
ENPP2 Q13822 1/20 0.32
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
GSK3B P49841 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12909893 1.00 NR1I2 (0.51) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL12949423 1.00 NR1I2 (0.51) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL12909589 0.95 NR1I2 (0.52) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL936718 0.93 NR1I2 (0.55) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL936716 0.93 NR1I2 (0.55) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL12909702 0.92 NR1I2 (0.54) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL12910162 0.92 NR1I2 (0.54) NR1I2CYP2E1MLNRENPP2BCHE
SCHEMBL12909798 0.91 CYP2E1 (0.54) NR1I2CYP2E1ENPP2BCHEACHE
SCHEMBL937903 0.91 CYP2E1 (0.54) NR1I2CYP2E1ENPP2BCHEACHE
SCHEMBL15354583 0.91 CYP2E1 (0.54) NR1I2CYP2E1ENPP2BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140030223-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES, INC. (US) 2014-01-30 US disclosed
US-8569302-B2 Inhibitors of flaviviridae viruses GILEAD SCIENCES, INC. (US) 2013-10-29 US disclosed
EP-2475657-B1 5-ALKINYLTHIEN-2-YLCARBOXYLIC ACIDS AS INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES INC (US) 2013-06-12 EP disclosed
US-20110020278-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES, INC. (US) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140030223-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES HAVCR2, CYP2F1, CYP4F3 NR1I2 88/4885CYP2E1 6/4885MLNR 3658/4885
US-20110020278-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES HAVCR2, CYP2F1, CYP4F3 NR1I2 88/4885CYP2E1 6/4885MLNR 3658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.