Travoprost

Travoprost

SCHEMBL93818

CC(C)OC(=O)CCC/C=C\C[C@@H]1[C@@H](/C=C/[C@@H](O)COc2cccc(C(F)(F)F)c2)[C@H](O)C[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGFR

The experimentally established mechanism targets of Travoprost. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGFR known ✓ P43088 14/20 1.00
ABCC4 O15439 2/20 1.00
ABCB11 O95342 2/20 1.00
PTGER3 P43115 4/20 0.81
TBXA2R P21731 4/20 0.64
PTGER1 P34995 2/20 0.63
THRB P10828 1/20 0.63
PTGER2 P43116 1/20 0.63
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Travoprost SCHEMBL10015920 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL11907120 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL2177084 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL10086843 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL15074545 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL2177092 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL20485616 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL20485617 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL20664855 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R
Travoprost SCHEMBL1951740 1.00 PTGFR (1.00) PTGFRABCC4ABCB11PTGER3TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11563 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107180-A1 IMPLANT INJECTOR DEVICE OCULAR THERAPEUTIX, INC. (US) 2026-05-21 WO claimed
EP-2308466-B2 Aqueous pharmaceutical compositions containing borate-polyol complexes NOVARTIS AG (CH) 2026-05-20 EP claimed
WO-2026102187-A1 ENGINEERED VIRUS-LIKE PARTICLES COMPRISING A BASE EDITOR FOR THE TREATMENT OF GLAUCOMA, AND APPLICATIONS THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-05-15 WO claimed
US-20260131008-A1 HYALURONIC ACID BASED DRUG DELIVERY SYSTEMS CELLA THERAPEUTICS LLC (US) 2026-05-14 US claimed
EP-4739302-A2 HYALURONIC ACID BASED DRUG DELIVERY SYSTEMS Cella Therapeutics, LLC (US) 2026-05-13 EP claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
EP-4727651-A1 METHOD OF ENHANCING THE SYSTEMIC HYPOGLYCEMIC EFFECT OF TOPICALLY APPLIED INSULIN WITH THE USE OF PROSTAGLANDIN ANALOGUES: A NOVEL FIXED COMBINATION EYE DROP FORMULATION OF INSULIN AND PROSTAGLANDIN ANALOGUE FOR THE LOWERING OF BLOOD GLUCOSE LEVEL Gosiengfiao, David Harold (PH) 2026-04-22 EP claimed
EP-3973954-B1 PRESERVATIVE FREE PHARMACEUTICAL COMPOSITIONS FOR OPHTHALMIC ADMINISTRATION NTC S R L (IT) 2026-04-22 EP claimed
EP-4724839-A2 CONTACT LENSES INCLUDING MEDICAMENTS AND METHODS OF MAKING AND USING SAME INCLUDING SLOW RELEASE OF GLAUCOMA TREATING DRUGS AND COMFORT ENHANCING DRUGS Mediprint Ophthalmics Inc. (US) 2026-04-15 EP claimed
EP-4724079-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION Stealth BioTherapeutics Inc. (US) 2026-04-15 EP claimed
WO-2002005815-A1 OPHTHALMIC FORMULATION OF A SELECTIVE CYCLOOXYGENASE-2 INHIBITORY DRUG PHARMACIA & UPJOHN COMPANY (US) 2002-01-24 WO claimed
EP-1169061-A1 COMBINATION THERAPY FOR TREATING GLAUCOMA ALCON LABORATORIES, INC. (US) 2002-01-09 EP claimed
WO-2001095913-A1 METHODS AND COMPOSITIONS FOR THE PREVENTION OF MYOPIA SYNPHORA AB (SE) 2001-12-20 WO claimed
US-20010047012-A1 COMBINATION THERAPY FOR TREATING GLAUCOMA ALCON RESEARCH, LTD. 2001-11-29 US claimed
US-20010023258-A1 Use of cloprostenol and fluprostenol analogues to treat glaucoma and ocular hypertension ALCON RESEARCH, LTD. 2001-09-20 US claimed
EP-1115406-A2 SUSTAINED RELEASE, AND COMFORTABLE OPHTHALMIC COMPOSITION AND METHOD FOR OCULAR THERAPY ALCON LABORATORIES, INC. (US) 2001-07-18 EP claimed
CN-1295483-A Gelling ophthalmic composition containing xanthan gum ALCON LAB INC (US) 2001-05-16 CN claimed
CN-1272063-A Prostaglandin product ALCON LAB INC (US) 2000-11-01 CN claimed
WO-2000054810-A1 COMBINATION THERAPY FOR TREATING GLAUCOMA ALCON LABORATORIES, INC (US) 2000-09-21 WO claimed
WO-2000018316-A2 SUSTAINED RELEASE, AND COMFORTABLE OPHTHALMIC COMPOSITION AND METHOD FOR OCULAR THERAPY ALCON LABORATORIES, INC. (US) 2000-04-06 WO claimed