SCHEMBL938799

SCHEMBL938799

O=CN(CCC1CCCCN1)c1cccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 14/20 0.51
BRAF P15056 3/20 0.47
KDR P35968 2/20 0.47
CDK8 P49336 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL938359 0.80 RAF1 (0.68) RAF1BRAFKDR
SCHEMBL13556629 0.71 RAF1 (0.72) RAF1BRAFKDRCDK8
SCHEMBL13529088 0.71 RAF1 (0.70) RAF1BRAFKDRCDK8
SCHEMBL13524681 0.70 RAF1 (0.74) RAF1BRAFKDRCDK8
SCHEMBL937746 0.70 RAF1 (0.65) RAF1BRAFKDRCDK8
SCHEMBL16628075 0.69 RAF1 (0.67) RAF1BRAFKDRCDK8
SCHEMBL16620784 0.69 KDR (0.73) RAF1BRAFKDRCDK8
SCHEMBL6014335 0.69 RAF1 (0.79) RAF1KDRCDK8
SCHEMBL19668099 0.68 RAF1 (0.80) RAF1BRAFKDRCDK8
Sc-43 SCHEMBL14684295 0.68 RAF1 (0.67) RAF1BRAFKDRCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324825-A1 Aryl ureas with angiogenesis inhibiting activity Bayer Healthcare LLC (US) 2011-05-25 EP claimed
EP-1478358-B1 Sorafenib tosylate for the treatment of diseases characterized by abnormal angiogenesis BAYER HEALTHCARE LLC (US) 2013-07-03 EP disclosed
EP-1636585-B2 DIARYL UREAS WITH KINASE INHIBITING ACTIVITY BAYER HEALTHCARE LLC (US) 2012-06-13 EP disclosed
EP-2324825-A1 Aryl ureas with angiogenesis inhibiting activity Bayer Healthcare LLC (US) 2011-05-25 EP disclosed
EP-2289515-A2 Combinations comprising a diaryl urea and an interferon Bayer HealthCare LLC (US) 2011-03-02 EP disclosed
US-20110015195-A1 ARYL UREAS WITH ANGIOGENISIS INHIBITING ACTIVITY DUMAS JACQUES 2011-01-20 US disclosed
US-7838541-B2 Aryl ureas with angiogenesis inhibiting activity BAYER HEALTHCARE, LLC (US) 2010-11-23 US disclosed
EP-1636585-B1 DIARYL UREAS WITH KINASE INHIBITING ACTIVITY BAYER PHARMACEUTICALS CORP (US) 2008-01-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110015195-A1 ARYL UREAS WITH ANGIOGENISIS INHIBITING ACTIVITY FLT1, FLT4, KDR RAF1 867/4885BRAF 487/4885KDR 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.