SCHEMBL9389830

SCHEMBL9389830

CCc1cccc2[nH]c(=O)c(O)cc(=O)c12

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DAO P14920 10/20 0.68
DDO Q99489 5/20 0.68
CDK1 P06493 1/20 0.44
CDK2 P24941 1/20 0.44
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9389414 0.90 DAO (0.58) DAODDOGRIN1GRIN2A
SCHEMBL16767853 0.81 DAO (1.00) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL8580170 0.81 DAO (0.66) DAODDO
SCHEMBL9389908 0.80 DAO (0.50) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL9389308 0.79 DAO (0.56) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL9389013 0.78 DAO (0.58) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL9389356 0.78 DAO (0.50) DAODDOCDK1CDK2
SCHEMBL9393158 0.78 DAO (0.66) DAODDOGRIN2DGRIN3BGRIN1
SCHEMBL9387612 0.78 DAO (0.66) DAODDO
SCHEMBL9392651 0.77 DAO (0.49) DAODDOCDK1CDK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994007500-A1 2,5-DIHYDRO-2,5-DIOXO-1H-AZEPINES AND 2,5-DIHYDRO-2-OXO-1H-AZEPINES AND THE USE THEREOF AS EXCITATORY AMINO ACID AND GLYCINE RECEPTOR ANTAGONISTS WEBER ECKARD (US) 1994-04-14 WO disclosed