SCHEMBL9401554

SCHEMBL9401554

COC(=O)C1=C(C)NC(C)=C(C(=O)OC/C=C/c2ccc(Cn3ccnc3)cc2)C1c1cccc(Cl)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 13/20 0.46
CYP2C9 P11712 3/20 0.46
CYP1A2 P05177 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
KMT2A Q03164 2/20 0.46
HIF1A Q16665 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ABCB11 O95342 2/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
TP53 P04637 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
THPO P40225 1/20 0.46
NR1I2 O75469 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401560 1.00 CACNA1B (0.46) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL9401689 0.93 CACNA1B (0.45) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL9401692 0.93 CACNA1B (0.45) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL7299355 0.92 CYP1A2 (0.56) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL7299361 0.92 CYP1A2 (0.56) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL9401866 0.92 CACNA1B (0.46) CACNA1BCYP1A2MEN1CYP3A4CYP2C19
SCHEMBL9401861 0.92 CACNA1B (0.46) CACNA1BCYP1A2MEN1CYP3A4CYP2C19
SCHEMBL9401555 0.89 CACNA1B (0.54) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL9401564 0.89 CACNA1B (0.54) CACNA1BCYP2C9CYP1A2KDM4EMEN1
SCHEMBL9401900 0.88 CACNA1B (0.48) CACNA1BCYP2C9CYP1A2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed