SCHEMBL9406597

SCHEMBL9406597

CCC[C@H]1CC[C@H](C(=O)Oc2ccc(OC(=O)[C@H]3CC[C@H](CCC)CC3)c(F)c2F)CC1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPGD P15428 4/20 0.40
MAPT P10636 3/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 2/20 0.39
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
F2 P00734 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9406600 1.00 CYP2C9 (0.40) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL7907306 0.95 HPGD (0.44) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL9562631 0.95 POLB (0.43) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL7907302 0.95 HPGD (0.44) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL9562624 0.95 POLB (0.43) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL9405776 0.92 HPGD (0.38) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL9405772 0.92 HPGD (0.38) CYP2C9KMT2AMEN1RAB9AL3MBTL1
SCHEMBL9405825 0.92 MAPT (0.46) KMT2AMEN1RAB9AL3MBTL1HPGD
SCHEMBL9405823 0.92 MAPT (0.46) KMT2AMEN1RAB9AL3MBTL1HPGD
SCHEMBL9562595 0.91 POLB (0.44) CYP2C9KMT2AMEN1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5279764-A Dihalogenobenzene derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-01-18 US disclosed
US-5248447-A 2,3-difluorohydroquinone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-09-28 US disclosed
EP-0332007-B1 DERIVATIVES OF 2,3-DIFLUOROHYDROQUINONE MERCK PATENT GmbH (DE) 1992-11-25 EP disclosed
EP-0373186-A1 DERIVATIVES OF 2,3-DIFLUOROHYDROQUINONE MERCK PATENT GmbH (DE) 1990-06-20 EP disclosed
WO-1989008637-A1 DERIVATIVES OF 2,3-DIFLUOROHYDROQUINONE MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-09-21 WO disclosed
EP-0332007-A1 Derivatives of 2,3-difluorohydroquinone MERCK PATENT GmbH (DE) 1989-09-13 EP disclosed