SCHEMBL9410375

SCHEMBL9410375

CC(C)(Cl)C(=O)c1cccc2c1NC(=O)CC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
GRM5 P41594 2/20 0.39
SMYD3 Q9H7B4 2/20 0.36
AHR P35869 1/20 0.36
KIF11 P52732 2/20 0.34
SRD5A1 P18405 2/20 0.34
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
KDM4E B2RXH2 2/20 0.33
POLB P06746 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP1A2 P05177 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9375230 0.77 AURKA (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL9529628 0.77 NPC1 (0.39) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL28629553 0.77 CRBN (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL7350316 0.77 NPC1 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL30114834 0.77 CRBN (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL6973213 0.74 PTPN1 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL1764695 0.70 AHR (0.70) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL2230502 0.70 NPC1 (0.50) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL29410901 0.70 NPC1 (0.50) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL434004 0.70 NPC1 (0.50) NPC1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579077-A2 1,3,4-Thiadiazinones for the treatment of cardiovascular diseases MERCK PATENT GmbH (DE) 1994-01-19 EP disclosed