SCHEMBL9417419

SCHEMBL9417419

CCC(C(=O)[O-])[N+](CC)(CC)CC

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.37
TSHR P16473 2/20 0.37
NFKB1 P19838 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
CA2 P00918 4/20 0.35
ALPL P05186 1/20 0.35
POLB P06746 1/20 0.35
ALPG P10696 1/20 0.35
BBOX1 O75936 3/20 0.33
CA1 P00915 2/20 0.32
FFAR3 O14843 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL2588435 0.78 TSHR (0.36) CYP3A4TSHRNFKB1NPSR1CA2
Ammonia Solution, Strong SCHEMBL9569011 0.78 CYP3A4 (0.32) CYP3A4TSHRNFKB1NPSR1CA2
SCHEMBL1427298 0.77 POLB (0.50) CYP3A4TSHRNFKB1NPSR1CA2
SCHEMBL10913359 0.76 MCL1 (0.32) CYP3A4TSHRNFKB1NPSR1ALPL
Ammonia Solution, Strong SCHEMBL6512029 0.76 TSHR (0.34) CYP3A4TSHRNFKB1NPSR1CA2
Hydrochloric Acid SCHEMBL25181737 0.75 POLB (0.48) CYP3A4TSHRNFKB1NPSR1CA2
SCHEMBL5322694 0.73 CYP3A4 (0.32) CYP3A4TSHRNFKB1NPSR1CA2
Acetic Acid SCHEMBL3682296 0.71 POLB (0.50) CYP3A4TSHRNFKB1NPSR1CA2
Acetic Acid SCHEMBL320011 0.70 CA1 (0.40) CYP3A4TSHRNFKB1NPSR1CA2
SCHEMBL15610744 0.65 CHRM1 (0.33) TSHRCA2ALPLPOLBALPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5373095-A Steroid compounds THE UPJOHN COMPANY (US) 1994-12-13 US disclosed
US-5334712-A Estrane or androstane pyridinyl alkyl or alkylphenyl amine steroids for antidiabetes and obesity THE UPJOHN COMPANY (US) 1994-08-02 US disclosed
US-5274089-A A estra-1,3,5(10)-triene derivative THE UPJOHN COMPANY (US) 1993-12-28 US disclosed
US-5196542-A Phospholipase A2 inhibitors THE UPJOHN COMPANY (US) 1993-03-23 US disclosed
US-5187299-A Phospholipase inhibitors; treating diabetes, obesity THE UPJOHN COMPANY (US) 1993-02-16 US disclosed
US-5145874-A Phospholipase inhibitor, hypoglycemic agent, antidiabetic, obesity THE UPJOHN COMPANY (US) 1992-09-08 US disclosed
US-4917826-A TREATING DIABETES AND OBESITY THE UPJOHN COMPANY (US) 1990-04-17 US disclosed