SCHEMBL9434183

SCHEMBL9434183

CC1=Nc2cc(Cl)ccc2Oc2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 1.00
HRH4 Q9H3N8 9/20 0.58
DRD4 P21917 6/20 0.58
DRD2 P14416 5/20 0.58
HRH2 P25021 3/20 0.48
HRH1 P35367 3/20 0.48
ADRA2A P08913 3/20 0.48
HTR2A P28223 3/20 0.48
ADRB2 P07550 2/20 0.48
CHRM2 P08172 2/20 0.48
CHRM4 P08173 2/20 0.48
HTR1A P08908 2/20 0.48
CHRM5 P08912 2/20 0.48
ADORA3 P0DMS8 2/20 0.48
CHRM1 P11229 2/20 0.48
ADRA2B P18089 2/20 0.48
ADRA2C P18825 2/20 0.48
CHRM3 P20309 2/20 0.48
DRD1 P21728 2/20 0.48
DRD5 P21918 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043895 0.87 MAPK1 (0.77) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL3254394 0.83 MAPK1 (0.71) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL123132 0.83 MAPK1 (0.71) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL1773258 0.81 MAPK1 (0.67) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL9434561 0.80 MAPK1 (0.67) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL9433516 0.78 MAPK1 (0.63) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL11097808 0.77 MAPK1 (0.62) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL11414467 0.75 MAPK1 (0.59) MAPK1HRH4DRD4DRD2HRH2
SCHEMBL12142524 0.74 MAPK1 (0.59) MAPK1HRH4DRD4DRD2HRH2
Iodide SCHEMBL11405476 0.74 MAPK1 (0.58) MAPK1HRH4DRD4DRD2HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5324722-A Analgesics G. D. SEARLE & CO. (US) 1994-06-28 US disclosed
WO-1993013082-A1 SUBSTITUTED DIBENZOXAZEPINES OR DIBENZOTHIAZEPINES AND THEIR USE AS PROSTAGLANDIN E2 ANTAGONISTS G.D. SEARLE & CO. (US) 1993-07-08 WO disclosed