SCHEMBL9440281

SCHEMBL9440281

COC(=O)[C@H](Cc1ccccc1)NC(=O)CCc1ccc(CP(=O)(O)O)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.56
HDAC6 Q9UBN7 5/20 0.56
PARP1 P09874 1/20 0.53
PARP3 Q9Y6F1 1/20 0.53
ATM Q13315 1/20 0.51
ALDH1A1 P00352 3/20 0.51
LMNA P02545 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
POLB P06746 1/20 0.51
HDAC8 Q9BY41 2/20 0.50
GLA P06280 1/20 0.50
MDM4 O15151 1/20 0.50
MDM2 Q00987 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5966500 0.89 HDAC1 (0.63) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL4145476 0.89 HDAC1 (0.63) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL4145473 0.89 HDAC1 (0.63) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL9556174 0.88 HDAC1 (0.53) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL4153061 0.85 MDM4 (0.67) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL4149820 0.85 MDM4 (0.67) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL4149824 0.85 MDM4 (0.67) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL4153058 0.85 MDM4 (0.67) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL9440111 0.84 HDAC1 (0.59) HDAC1HDAC6PARP1PARP3ATM
SCHEMBL9440106 0.84 HDAC1 (0.59) HDAC1HDAC6PARP1PARP3ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526488-B1 BENZYLPHOSPHONIC ACID TYROSINE KINASE INHIBITORS PFIZER (US) 1994-11-30 EP disclosed
US-5326905-A Benzylphosphonic acid tyrosine kinase inhibitors PFIZER INC. (US) 1994-07-05 US disclosed
WO-1991015495-A1 BENZYLPHOSPHONIC ACID TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1991-10-17 WO disclosed