SCHEMBL9440328

SCHEMBL9440328

CC1(COc2ccc(CBr)cc2)CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.53
TSHR P16473 3/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAPT P10636 1/20 0.53
ALOX15 P16050 1/20 0.53
KMT2A Q03164 1/20 0.53
HSD17B10 Q99714 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
PARP1 P09874 1/20 0.50
PPARG P37231 1/20 0.43
ACACB O00763 2/20 0.40
HRH3 Q9Y5N1 5/20 0.33
PSMB1 P20618 2/20 0.32
PSMB5 P28074 2/20 0.32
PSMB2 P49721 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL508167 0.83 HPGD (0.53) HPGDTSHRMEN1ALDH1A1TP53
Hydrochloric Acid SCHEMBL507244 0.82 HPGD (0.52) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL9440408 0.81 HPGD (0.54) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL8503886 0.79 HPGD (0.52) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL9440267 0.77 HPGD (0.54) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL1299701 0.75 HPGD (0.63) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL507935 0.74 HPGD (0.51) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL9440366 0.74 HPGD (0.48) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL19023278 0.74 HPGD (0.47) HPGDTSHRMEN1ALDH1A1TP53
SCHEMBL18072 0.73 HPGD (0.46) HPGDTSHRMEN1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526488-B1 BENZYLPHOSPHONIC ACID TYROSINE KINASE INHIBITORS PFIZER (US) 1994-11-30 EP disclosed
US-5326905-A Benzylphosphonic acid tyrosine kinase inhibitors PFIZER INC. (US) 1994-07-05 US disclosed
EP-0526488-A1 BENZYLPHOSPHONIC ACID TYROSINE KINASE INHIBITORS. PFIZER (US) 1993-02-10 EP disclosed
WO-1991015495-A1 BENZYLPHOSPHONIC ACID TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1991-10-17 WO disclosed