SCHEMBL9455459

SCHEMBL9455459

Cc1c(F)c(N2CCNC(C(=O)O)C2)cc2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.83
HRH3 Q9Y5N1 1/20 0.83
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 4/20 0.51
HPGD P15428 3/20 0.51
HSD17B10 Q99714 3/20 0.51
TOP2A P11388 3/20 0.51
TOP2B Q02880 3/20 0.51
LMNA P02545 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPT P10636 1/20 0.44
POLB P06746 2/20 0.44
PRKD3 O94806 1/20 0.44
ALOX15 P16050 1/20 0.44
OPRM1 P35372 1/20 0.44
CLK2 P49760 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Grepafloxacin SCHEMBL34155 0.91 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL34156 0.91 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL34157 0.91 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL29695614 0.91 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL2636690 0.90 KCNH2 (0.98) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL1230941 0.90 KCNH2 (0.98) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL29419670 0.90 KCNH2 (0.98) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL7763536 0.90 KCNH2 (0.98) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL137804 0.90 KCNH2 (0.98) KCNH2HRH3KDM4EALDH1A1HPGD
Grepafloxacin SCHEMBL7763531 0.90 KCNH2 (0.98) KCNH2HRH3KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5078326-A None JP disclosed
JP-H0578326-A BENZOHETEROCYCLIC COMPOUND OTSUKA PHARMACEUT CO LTD 1993-03-30 JP disclosed
JP-H00578326-A 0001-01-01 JP disclosed