SCHEMBL9458436

SCHEMBL9458436

Cc1cccc(CCOc2ccc(CC3SC(=N)NC3=O)cc2)n1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARG P37231 13/20 0.53
CYP3A4 P08684 1/20 0.52
RXRA P19793 1/20 0.52
MAOB P27338 1/20 0.51
FFAR1 O14842 7/20 0.43
ESR1 P03372 1/20 0.42
PPARA Q07869 1/20 0.42
MPC2 O95563 2/20 0.42
CYP2C8 P10632 2/20 0.42
CYP2C9 P11712 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196242 0.89 PPARG (0.66) PPARGCYP3A4RXRAFFAR1PPARA
SCHEMBL9458269 0.87 PPARG (0.52) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL14519307 0.84 MAOB (0.57) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL5172074 0.82 PPARG (0.64) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL2944577 0.80 PPARG (0.80) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL30640947 0.80 PPARG (0.80) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL13475125 0.80 PPARG (0.80) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL12521693 0.79 PPARG (0.64) PPARGCYP3A4RXRAFFAR1PPARA
Hydrochloric Acid SCHEMBL1162844 0.79 PPARG (0.81) PPARGCYP3A4RXRAMAOBFFAR1
SCHEMBL9458054 0.79 MAOB (0.51) PPARGCYP3A4RXRAMAOBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5183823-A PYRIDINE N-OXIDE COMPOUNDS WHICH ARE USEFUL AS HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-02-02 US disclosed