SCHEMBL9485698

SCHEMBL9485698

CCC(F)CC[C@H]1CC[C@H](c2ccc(C#N)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.43
GRIA2 P42262 1/20 0.43
GRIA3 P42263 1/20 0.43
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP2C9 P11712 1/20 0.39
HSD11B1 P28845 1/20 0.38
USP30 Q70CQ3 4/20 0.38
ESR2 Q92731 2/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HRH3 Q9Y5N1 2/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
KDM1A O60341 2/20 0.35
KCNH2 Q12809 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9485694 1.00 GRIA1 (0.43) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL9326560 0.87 GRIA1 (0.42) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL9326567 0.87 GRIA1 (0.42) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL11618153 0.86 GRIA2 (0.45) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL9450875 0.84 GRIA1 (0.48) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL1658450 0.82 MEN1 (0.56) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL261024 0.82 MEN1 (0.56) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL9325765 0.82 GRIA1 (0.41) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL9325768 0.82 GRIA1 (0.41) GRIA1GRIA2GRIA3MEN1MAPK1
SCHEMBL10832031 0.81 MEN1 (0.55) GRIA1GRIA2GRIA3MEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252252-A Longitudinal polarization MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1993-10-12 US disclosed
US-5230829-A PHENYLCYCLOHEXANES, AND A LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-07-27 US disclosed
US-5120467-A Longitudinal polarization and-or cross-polarization MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-06-09 US disclosed
EP-0478740-A1 PHENYL CYCLOHEXANES AND LIQUID CRYSTALLINE MEDIUM MERCK PATENT GmbH (DE) 1992-04-08 EP disclosed
WO-1991016291-A1 PHENYL CYCLOHEXANES AND LIQUID CRYSTALLINE MEDIUM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-10-31 WO disclosed
US-4723005-A CONTAINING POLARIZED CYANO OR HALOGEN SUBSTITUENTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1988-02-02 US disclosed
EP-0139996-B1 ANISOTROPIC COMPOUNDS AND LIQUID CRYSTAL MIXTURES MERCK PATENT GmbH (DE) 1987-11-04 EP disclosed
EP-0139996-A1 Anisotropic compounds and liquid crystal mixtures MERCK PATENT GmbH (DE) 1985-05-08 EP disclosed