SCHEMBL949147

SCHEMBL949147

O=C(O)/C=C/c1cc2cc(OCc3ccccc3)ccc2n1CCO

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.55
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
PKM P14618 1/20 0.53
PTGER3 P43115 1/20 0.51
PTGDR Q13258 1/20 0.51
MEN1 O00255 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 1/20 0.50
LTB4R Q15722 2/20 0.47
LTB4R2 Q9NPC1 2/20 0.47
ALOX5 P09917 1/20 0.45
F10 P00742 1/20 0.44
MAOB P27338 1/20 0.43
GSK3B P49841 1/20 0.43
BACE1 P56817 1/20 0.43
P2RY14 Q15391 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949148 1.00 SRD5A2 (0.55) SRD5A2ALDH1A1KDM4EPKMPTGER3
SCHEMBL949755 0.87 SRD5A2 (0.52) SRD5A2MEN1NPC1RAB9AKMT2A
SCHEMBL949756 0.87 SRD5A2 (0.52) SRD5A2MEN1NPC1RAB9AKMT2A
SCHEMBL946360 0.87 SRD5A2 (0.51) SRD5A2ALDH1A1KDM4EPKMMEN1
SCHEMBL946357 0.87 SRD5A2 (0.51) SRD5A2ALDH1A1KDM4EPKMMEN1
SCHEMBL8131616 0.85 PTGER3 (0.50) SRD5A2ALDH1A1KDM4EPKMPTGER3
SCHEMBL8150530 0.85 PTGER3 (0.50) SRD5A2ALDH1A1KDM4EPKMPTGER3
SCHEMBL7246674 0.85 PTGER3 (0.55) SRD5A2ALDH1A1KDM4EPKMPTGER3
SCHEMBL7246667 0.85 PTGER3 (0.55) SRD5A2ALDH1A1KDM4EPKMPTGER3
SCHEMBL945581 0.84 SRD5A2 (0.51) SRD5A2ALDH1A1KDM4EPKMPTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed