SCHEMBL9494975

SCHEMBL9494975

CCCOc1ccc(C#Cc2cnc(C#Cc3ccc(OCCC)cc3)nc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.53
ACACB O00763 14/20 0.47
LTA4H P09960 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9495676 0.93 MCHR1 (0.53) MCHR1ACACBLTA4HCHRNB2CHRNB4
SCHEMBL9498090 0.90 KDM4E (0.52) MCHR1ACACBLTA4H
SCHEMBL9495615 0.90 MCHR1 (0.51) MCHR1ACACBLTA4HCHRNB2CHRNB4
SCHEMBL9495038 0.89 KDM4E (0.55) MCHR1LTA4H
SCHEMBL9495779 0.89 KDM4E (0.55) MCHR1LTA4H
SCHEMBL9497471 0.89 NPC1 (0.53) MCHR1ACACBLTA4HCHRNB2CHRNB4
SCHEMBL9496054 0.89 MCHR1 (0.50) MCHR1ACACB
SCHEMBL9496057 0.89 KDM4E (0.55) MCHR1LTA4H
SCHEMBL9497455 0.87 MCHR1 (0.49) MCHR1ACACB
SCHEMBL9854862 0.86 NQO1 (0.52) MCHR1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed