SCHEMBL9495658

SCHEMBL9495658

CC[C@H]1CC[C@H](c2ccc(C#Cc3ncc(OC)cn3)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.43
ACACB O00763 3/20 0.37
DRD2 P14416 1/20 0.36
EGLN1 Q9GZT9 1/20 0.34
EGLN3 Q9H6Z9 1/20 0.34
NPBWR1 P48145 1/20 0.34
RAB9A P51151 1/20 0.32
APP P05067 2/20 0.32
GRM2 Q14416 1/20 0.32
KDM1A O60341 1/20 0.31
GRM3 Q14832 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9495667 1.00 MCHR1 (0.43) MCHR1ACACBDRD2EGLN1EGLN3
SCHEMBL9496093 0.90 CYP2C9 (0.42) MCHR1ACACBDRD2EGLN1EGLN3
SCHEMBL9496084 0.90 CYP2C9 (0.42) MCHR1ACACBDRD2EGLN1EGLN3
SCHEMBL9496182 0.90 ACACB (0.44) MCHR1ACACBEGLN1EGLN3
SCHEMBL9496173 0.90 ACACB (0.44) MCHR1ACACBEGLN1EGLN3
SCHEMBL9497472 0.88 MCHR1 (0.40) MCHR1ACACBDRD2EGLN1EGLN3
SCHEMBL9497477 0.88 MCHR1 (0.40) MCHR1ACACBDRD2EGLN1EGLN3
SCHEMBL9497565 0.88 MCHR1 (0.39) MCHR1ACACBRAB9A
SCHEMBL9497557 0.88 MCHR1 (0.39) MCHR1ACACBRAB9A
SCHEMBL9497397 0.87 ESR2 (0.41) MCHR1ACACBDRD2EGLN1EGLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed
EP-0306505-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES. MERCK PATENT GMBH (DE) 1989-03-15 EP disclosed
WO-1988007523-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed