SCHEMBL9495945

SCHEMBL9495945

CCC[C@H]1CC[C@H](C#Cc2ccc(-c3ccc(C#N)cc3)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KIF11 P52732 2/20 0.39
FFAR1 O14842 1/20 0.38
HRH2 P25021 3/20 0.36
HRH1 P35367 3/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9495948 1.00 HRH3 (0.40) HRH3TSHRHSD17B10KIF11FFAR1
SCHEMBL10513390 0.96 HRH3 (0.38) HRH3TSHRHSD17B10KIF11FFAR1
SCHEMBL9498022 0.92 TSHR (0.44) HRH3TSHRHSD17B10KIF11FFAR1
SCHEMBL9498026 0.92 TSHR (0.44) HRH3TSHRHSD17B10KIF11FFAR1
SCHEMBL9499565 0.91 FFAR1 (0.38) HRH3FFAR1
SCHEMBL9855252 0.91 FFAR1 (0.38) HRH3FFAR1
SCHEMBL9499571 0.91 FFAR1 (0.38) HRH3FFAR1
SCHEMBL9497569 0.91 TSHR (0.47) HRH3TSHRHSD17B10KIF11FFAR1
SCHEMBL9497566 0.91 TSHR (0.47) HRH3TSHRHSD17B10KIF11FFAR1
SCHEMBL9495306 0.89 TSHR (0.49) HRH3TSHRHSD17B10KIF11FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed