SCHEMBL9496105

SCHEMBL9496105

CCCCOc1ccc(C#Cc2ccc(C)cn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.50
ACACB O00763 4/20 0.47
GRM5 P41594 1/20 0.43
CYP2D6 P10635 4/20 0.43
CHRM1 P11229 2/20 0.43
HTR2A P28223 2/20 0.43
CYP3A4 P08684 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 2/20 0.41
CYP19A1 P11511 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9496274 0.97 MCHR1 (0.48) MCHR1ACACBGRM5CYP2D6CHRM1
SCHEMBL9497983 0.96 MCHR1 (0.47) MCHR1ACACB
SCHEMBL9500610 0.96 MCHR1 (0.47) MCHR1ACACB
SCHEMBL9496650 0.96 MCHR1 (0.47) MCHR1ACACB
SCHEMBL9495680 0.94 ACACB (0.53) MCHR1ACACBGRM5CYP2D6CHRM1
SCHEMBL9500659 0.89 MCHR1 (0.53) MCHR1ACACBCYP2D6CHRM1HTR2A
SCHEMBL9495556 0.88 ACACB (0.54) MCHR1ACACBGRM5
SCHEMBL9497308 0.86 KDM4E (0.51) MCHR1ACACBCYP2D6CHRM1HTR2A
SCHEMBL9497336 0.84 ACACB (0.52) MCHR1ACACBCYP2D6CHRM1HTR2A
SCHEMBL9496092 0.84 MCHR1 (0.54) MCHR1ACACBCYP2D6CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed