SCHEMBL9501959

SCHEMBL9501959

CC(=O)c1ccc(Cl)c(Cl)c1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.39
CYP3A4 P08684 2/20 0.39
DPP4 P27487 1/20 0.39
NOTUM Q6P988 3/20 0.38
TSHR P16473 2/20 0.38
HPGD P15428 3/20 0.37
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
NSD2 O96028 1/20 0.37
POLB P06746 1/20 0.37
MCL1 Q07820 1/20 0.37
CASP1 P29466 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CXCR1 P25024 1/20 0.37
CXCR2 P25025 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
TDP1 Q9NUW8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14882745 0.84 DPP4 (0.45) MAPK1CYP3A4DPP4TSHRHPGD
SCHEMBL4509639 0.83 DPP4 (0.43) MAPK1CYP3A4DPP4NOTUMTSHR
SCHEMBL481034 0.83 MAPT (0.44) MAPK1CYP3A4HPGDMAPTALDH1A1
SCHEMBL403103 0.82 CYP3A4 (0.42) MAPK1CYP3A4NOTUMTSHRMAPT
SCHEMBL30610932 0.82 CYP3A4 (0.42) MAPK1CYP3A4NOTUMTSHRMAPT
SCHEMBL21822958 0.81 MAPT (0.38) MAPK1CYP3A4HPGDMAPTALDH1A1
SCHEMBL18542465 0.81 TSHR (0.45) DPP4TSHRHPGDMAPTALDH1A1
SCHEMBL30084375 0.80 TSHR (0.54) DPP4TSHRHPGDMAPTALDH1A1
SCHEMBL73043 0.80 TSHR (0.54) DPP4TSHRHPGDMAPTALDH1A1
SCHEMBL1901357 0.79 MAOB (0.42) MAPK1CYP3A4HPGDMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110511233-B Thiazolo [2,3-b ] oxazolone compound and preparation method and application thereof 成都大学 2022-01-25 CN disclosed
EP-0305952-B1 SUBSTITUTED 2-PHENYL-4-QUINOLINE-CARBOXYLIC ACIDS AMERICAN CYANAMID COMPANY (US) 1993-06-02 EP disclosed
US-4847381-A ANTIARTHRITIC AGENTS AMERICAN CYANAMID COMPANY (US) 1989-07-11 US disclosed
EP-0305952-A1 Substituted 2-phenyl-4-quinoline-carboxylic acids AMERICAN CYANAMID COMPANY (US) 1989-03-08 EP disclosed