SCHEMBL9501983

SCHEMBL9501983

O=C(O)c1c(O)c(-c2ccc(Cl)cc2)nc2ccc(I)cc12

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 20/20 0.74
CYP3A4 P08684 2/20 0.54
CYP2C8 P10632 2/20 0.54
CYP2C9 P11712 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2A6 P11509 1/20 0.54
CYP2C19 P33261 1/20 0.54
PDE10A Q9Y233 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9505820 0.92 DHODH (0.63) DHODHPDE10A
SCHEMBL27434750 0.90 DHODH (0.60) DHODHCYP3A4CYP2C8CYP2C9CYP1A2
SCHEMBL9502241 0.89 DHODH (0.82) DHODHCYP3A4CYP2C8CYP2C9CYP1A2
SCHEMBL9502003 0.87 DHODH (0.70) DHODHPDE10A
SCHEMBL10583075 0.85 DHODH (1.00) DHODHCYP3A4CYP2C8CYP2C9CYP1A2
SCHEMBL10582725 0.84 DHODH (1.00) DHODH
SCHEMBL10582434 0.84 DHODH (1.00) DHODHCYP3A4CYP2C8CYP2C9CYP1A2
SCHEMBL10584241 0.83 DHODH (0.76) DHODHPDE10A
SCHEMBL9501955 0.81 DHODH (0.81) DHODHCYP3A4CYP2C8CYP2C9CYP1A2
SCHEMBL8793778 0.79 DHODH (0.58) DHODHCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0305952-B1 SUBSTITUTED 2-PHENYL-4-QUINOLINE-CARBOXYLIC ACIDS AMERICAN CYANAMID COMPANY (US) 1993-06-02 EP disclosed
US-4847381-A ANTIARTHRITIC AGENTS AMERICAN CYANAMID COMPANY (US) 1989-07-11 US disclosed
EP-0305952-A1 Substituted 2-phenyl-4-quinoline-carboxylic acids AMERICAN CYANAMID COMPANY (US) 1989-03-08 EP disclosed