SCHEMBL9505698

SCHEMBL9505698

Nc1nc(Cl)nc2c1ncn2C(=O)C(F)(F)[C@H](O)[C@H](O)CO

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.41
CFTR P13569 1/20 0.41
ADORA3 P0DMS8 6/20 0.39
ADORA2A P29274 4/20 0.39
ADORA1 P30542 3/20 0.39
PDE4D Q08499 2/20 0.39
PDE3A Q14432 2/20 0.39
PDE2A O00408 1/20 0.39
ADRA1A P35348 1/20 0.39
NT5E P21589 3/20 0.37
CD99 P14209 1/20 0.37
PNP P00491 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
HSP90B1 P14625 3/20 0.36
CHKA P35790 2/20 0.36
HSP90AA1 P07900 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9167926 0.89 CDK1 (0.42) CDK1ADORA3ADORA2AADORA1HSP90B1
SCHEMBL9141840 0.87
SCHEMBL8972502 0.83 GSK3B (0.51) ADORA2AADORA1
SCHEMBL8743023 0.83 GSK3B (0.51) ADORA2AADORA1
SCHEMBL8742970 0.83 GSK3B (0.51) ADORA2AADORA1
SCHEMBL8743090 0.79 BLM (0.48) PDE3APNPLMNASMN1; SMN2
SCHEMBL9139603 0.79 HPGD (0.41) PDE3ANT5EPNPLMNASMN1; SMN2
SCHEMBL8742956 0.79 BLM (0.48) PDE3APNPLMNASMN1; SMN2
SCHEMBL8742951 0.79 BLM (0.48) PDE3APNPLMNASMN1; SMN2
SCHEMBL8743135 0.72 TET2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0184365-B1 IMPROVEMENTS IN THE TREATMENT OF TUMORS IN MAMMALS ELI LILLY AND COMPANY (US) 1993-08-04 EP claimed
EP-0184365-A2 Improvements in the treatment of tumors in mammals ELI LILLY AND COMPANY (US) 1986-06-11 EP claimed