SCHEMBL9508456

SCHEMBL9508456

O=C(C(Cl)Cl)N1CCc2ccccc2C1c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 3/20 0.57
CYP2D6 P10635 1/20 0.56
CHRM3 P20309 4/20 0.53
CHRM2 P08172 2/20 0.53
CHRM1 P11229 2/20 0.53
CACNA1F O60840 1/20 0.53
CHRM4 P08173 1/20 0.53
CHRM5 P08912 1/20 0.53
KCNE1 P15382 1/20 0.53
KCNQ1 P51787 1/20 0.53
CACNA1D Q01668 1/20 0.53
KCNH2 Q12809 1/20 0.53
CACNA1S Q13698 1/20 0.53
CACNA1C Q13936 1/20 0.53
SCN5A Q14524 1/20 0.53
KCND3 Q9UK17 1/20 0.53
PRCP P42785 2/20 0.52
HDAC8 Q9BY41 2/20 0.51
TRPM8 Q7Z2W7 2/20 0.50
HDAC3 O15379 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509161 0.89 HHAT (0.61) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL29924098 0.84 HHAT (0.57) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL1567224 0.84 HHAT (0.57) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL1567218 0.84 HHAT (0.57) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL12153444 0.84 HHAT (0.57) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL12226990 0.84 HHAT (0.60) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL1122195 0.84 HHAT (0.60) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL698295 0.84 HHAT (0.60) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL15598479 0.84 TRPV1 (0.63) HHATCYP2D6CHRM3CHRM2CHRM1
SCHEMBL4250247 0.84 HHAT (0.60) HHATCYP2D6CHRM3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP claimed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP claimed
EP-0230871-B1 HALOACYL 1-SUBSTITUTED-1,2,3,4-TETRAHYDROISOQUINOLINES AS HERBICIDE ANTIDOTES Monsanto Company (US) 1993-09-22 EP disclosed
US-4755218-A Reducing acetochlor injury to corn by applying with antidote MONSANTO COMPANY (US) 1988-07-05 US disclosed
EP-0230871-A2 Haloacyl 1-substituted-1,2,3,4-tetrahydroisoquinolines as herbicide antidotes Monsanto Company (US) 1987-08-05 EP disclosed