SCHEMBL9512484

SCHEMBL9512484

COc1ccc(C#Cc2ccc(-c3ccc(C)cc3)cc2)c(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.44
AR P10275 3/20 0.37
ACHE P22303 1/20 0.35
GRM5 P41594 2/20 0.35
CA12 O43570 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
KCNH2 Q12809 2/20 0.35
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
CA1 P00915 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
FFAR1 O14842 1/20 0.33
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91913 0.97 AAK1 (0.43) AAK1ARACHEGRM5CA12
SCHEMBL10448649 0.91 AAK1 (0.40) AAK1ARACHEGRM5CA12
SCHEMBL9512496 0.85 AAK1 (0.38) AAK1ARGRM5CA12CA2
SCHEMBL9512290 0.84 FFAR1 (0.39) AAK1FFAR1MCHR1
SCHEMBL9508826 0.81 AAK1 (0.36) AAK1CA12CA2CA9KCNH2
SCHEMBL9511390 0.81 FFAR1 (0.42) AAK1FFAR1MCHR1
SCHEMBL9509326 0.81 AR (0.37) AAK1ARGRM5CA12CA2
SCHEMBL12994542 0.81 AAK1 (0.39) AAK1ACHEGRM5KDM4ENPC1
SCHEMBL9509953 0.80 CYP2D6 (0.37) AAK1KCNH2MCHR1
SCHEMBL4567628 0.80 GRM5 (0.39) AAK1ARACHEGRM5CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP disclosed