SCHEMBL9515046

SCHEMBL9515046

N[C@@H]1Cc2ccc3ccccc3c2C[C@H]1O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 3/20 0.53
KDM1A O60341 1/20 0.39
DPP4 P27487 2/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
RCE1 Q9Y256 1/20 0.38
HSD17B10 Q99714 2/20 0.35
CYP2A6 P11509 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HIF1A Q16665 1/20 0.35
CYP1B1 Q16678 1/20 0.35
NPY5R Q15761 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9515057 1.00 ANPEP (0.53) ANPEPKDM1ADPP4ALDH1A1KDM4E
SCHEMBL9515050 1.00 ANPEP (0.53) ANPEPKDM1ADPP4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9516290 0.98 ANPEP (0.51) ANPEPKDM1ADPP4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9516294 0.98 ANPEP (0.51) ANPEPKDM1ADPP4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9516301 0.98 ANPEP (0.51) ANPEPKDM1ADPP4ALDH1A1KDM4E
SCHEMBL6990855 0.73 KDM4E (0.57) ANPEPALDH1A1KDM4EGLAGAA
SCHEMBL11355392 0.72 ANPEP (0.68) ANPEP
SCHEMBL9515317 0.72 ANPEP (0.68) ANPEP
SCHEMBL3996873 0.72 ANPEP (0.68) ANPEP
SCHEMBL30070669 0.72 ANPEP (0.68) ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0378456-B1 TETRALIN DERIVATIVES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-15 EP disclosed
US-5106861-A Method of using certain tetralin derivatives to produce analgesic relief MERRELL DOW PHARMACEUTICALS INC. (US) 1992-04-21 US disclosed
US-5041673-A Aminopeptidase inhibitors, immunomodulators, analgesics MERRELL DOW PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed
EP-0378456-A1 Tetralin derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1990-07-18 EP disclosed