SCHEMBL9518044

SCHEMBL9518044

OC(c1ccccc1Br)C1CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A3 Q16572 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
PDE2A O00408 1/20 0.42
OPRL1 P41146 3/20 0.36
CFTR P13569 2/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
HTT P42858 1/20 0.34
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
NR1I2 O75469 1/20 0.33
HSD11B1 P28845 1/20 0.33
CYP3A4 P08684 2/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744668 1.00 SLC18A3 (0.44) SLC18A3SIGMAR1PDE2AOPRL1CFTR
SCHEMBL6745262 1.00 SLC18A3 (0.44) SLC18A3SIGMAR1PDE2AOPRL1CFTR
SCHEMBL14830564 0.81 PDE2A (0.41) SLC18A3SIGMAR1PDE2AOPRK1NR1I2
SCHEMBL1017887 0.81 SLC18A3 (0.35) SLC18A3SIGMAR1OPRL1CFTR
SCHEMBL2479070 0.75 HTT (0.38) SLC18A3SIGMAR1OPRL1IDO1TDO2
SCHEMBL2472871 0.75 HTT (0.38) SLC18A3SIGMAR1OPRL1IDO1TDO2
SCHEMBL4610704 0.75 ESR1 (0.43) PDE2AOPRL1IDO1TDO2OPRM1
SCHEMBL2504578 0.75 OPRL1 (0.45) PDE2AOPRL1IDO1TDO2OPRM1
SCHEMBL4610755 0.75 ESR1 (0.43) PDE2AOPRL1IDO1TDO2OPRM1
SCHEMBL5485147 0.75 PDE2A (0.54) PDE2AOPRL1IDO1TDO2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022040157-A1 BORON CONTAINING COMPOUNDS AND THEIR USES 5METIS, INC. (US) 2022-02-24 WO disclosed
WO-2022040157-A1 BORON CONTAINING COMPOUNDS AND THEIR USES 5METIS, INC. (US) 2022-02-24 WO disclosed
EP-0559743-A1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE. PFIZER HOSPITAL PROD (US) 1993-09-15 EP disclosed
WO-1992009566-A1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE PFIZER INC. (US) 1992-06-11 WO disclosed