Sb-203580

Sb-203580

SCHEMBL95208

C[S+]([O-])c1ccc(-c2nc(-c3ccc(F)cc3)c(-c3ccncc3)[nH]2)cc1

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 16/20 0.75
MAPK14 Q16539 16/20 0.75
MAPK13 O15264 15/20 0.75
MAPK12 P53778 15/20 0.75
GCGR P47871 14/20 0.75
CSNK1A1 P48729 5/20 0.75
CSNK1D P48730 5/20 0.75
PRKD3 O94806 4/20 0.75
MAP4K4 O95819 4/20 0.75
FRK P42685 4/20 0.75
MAPK9 P45984 4/20 0.75
GSK3B P49841 4/20 0.75
CLK4 Q9HAZ1 3/20 0.75
PTK6 Q13882 3/20 0.75
PRKD2 Q9BZL6 3/20 0.75
ALOX5 P09917 13/20 0.68
ALDH1A1 P00352 4/20 0.67
CSNK1E P49674 3/20 0.67
CSNK1A1L Q8N752 3/20 0.67
PRKACA P17612 3/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9192799 1.00 MAPK11 (0.75) MAPK11MAPK14MAPK13MAPK12GCGR
Sb-203580 SCHEMBL27075368 1.00 MAPK11 (0.75) MAPK11MAPK14MAPK13MAPK12GCGR
Sb-203580 SCHEMBL220990 1.00 MAPK11 (0.75) MAPK11MAPK14MAPK13MAPK12GCGR
Sb-203580 SCHEMBL25800837 1.00 MAPK11 (0.75) MAPK11MAPK14MAPK13MAPK12GCGR
Sb-203580 SCHEMBL146399 1.00 MAPK11 (0.75) MAPK11MAPK14MAPK13MAPK12GCGR
Sb-203580 SCHEMBL4890447 0.99 MAPK11 (0.73) MAPK11MAPK14MAPK13MAPK12GCGR
SCHEMBL20335254 0.90 MAPK11 (0.79) MAPK11MAPK14MAPK13MAPK12GCGR
SCHEMBL6447875 0.89 MAPK13 (0.72) MAPK11MAPK14MAPK13MAPK12GCGR
SCHEMBL1389121 0.87 MAPK14 (0.67) MAPK11MAPK14MAPK13MAPK12GCGR
SCHEMBL6606221 0.87 MAPK11 (0.70) MAPK11MAPK14MAPK13MAPK12GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2797 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260132384-A1 METHOD FOR REPROGRAMMING HUMAN SOMATIC CELLS INTO INDUCED PLURIPOTENT STEM CELLS EXONEUGLIA BIOTECHNOLOGY (SUZHOU) CO., LTD. (CN) 2026-05-14 US claimed
EP-4741496-A1 METHOD FOR REPROGRAMMING HUMAN SOMATIC CELLS INTO INDUCED PLURIPOTENT STEM CELLS Exoneuglia Biotechnology (Suzhou) Co., Ltd. (CN) 2026-05-13 EP claimed
US-20260109951-A1 METHODS AND COMPOSITIONS FOR INDUCING HEMATOPOIETIC CELL DIFFERENTIATION FATE THERAPEUTICS INC (US) 2026-04-23 US claimed
EP-4720261-A1 NOVEL CULTURE CONDITIONS FOR CLONAL EXPANSION OF NEPHRON PROGENITOR CELLS, GENERATION OF NEPHRON ORGANOIDS, AND RAPID AND SCALABLE MODELING OF POLYCYSTIC KIDNEY DISEASE University of Southern California (US) 2026-04-08 EP claimed
US-20260022341-A1 METHOD OF GENERATING A HOMOCELLULAR PROGENITOR CELL CULTURE FROM A HETEROCELLULAR TISSUE SAMPLE Mosa Meat B.V. (NL) 2026-01-22 US claimed
US-20260015632-A1 CULTURE MEDIUM COMBINATION FOR INDUCING DIFFERENTIATION OF PLURIPOTENT STEM CELLS INTO CD34+ HEMATOPOIETIC STEM/PROGENITOR CELLS SHENZHEN CELL INSPIRE BIOTECHNOLOGY CO., LTD. (CN) 2026-01-15 US claimed
EP-4665845-A1 PLURIPOTENT STEM CELL-ENGINEERED IMMUNE CELLS FOR OFF-THE-SHELF CELL THERAPY The Regents of University of California (US) 2025-12-24 EP claimed
US-12503685-B2 Cortical interneurons and other neuronal cells produced by the directed differentiation of pluripotent and multipotent cells MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2025-12-23 US claimed
US-20250340848-A1 METHODS FOR CHEMICAL REPROGRAMMING AND PLURIPOTENT STEM CELLS PEKING UNIVERSITY (CN) 2025-11-06 US claimed
EP-4640238-A1 THERAPEUTIC AGENT FOR PULMONARY DISEASE, HEPATIC DISEASE OR RENAL DISEASE, WHICH CONTAINS PGAM-CHK1 BINDING INHIBITOR Kyoto University (JP) 2025-10-29 EP claimed
US-20020028798-A1 Irrigation solution and method for inhibition of pain and inflammation OMEROS MEDICAL SYSTEMS 2002-03-07 US claimed
US-6288089-B1 ADMINISTERING A COMPOSITION OF PYRIDYL IMIDAZOLE COMPOUNDS TO TREAT PARKINSON'S DISEASE, HUNTINGTON'S DISEASE, ALZHEIMER'S DISEASE, AND AMYOTOPHIC LATERAL SCLEROSIS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2001-09-11 US claimed
US-6235760-B1 CENTRAL NERVOUS SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS SMITHKLINE BEECHAM CORPORATION 2001-05-22 US claimed
WO-2001019322-A2 USE OF CSAIDS IN RHINOVIRUS INFECTION SMITHKLINE BEECHAM CORPORATION (US) 2001-03-22 WO claimed
WO-2000023072-A1 IRRIGATION SOLUTION CONTAINING MAPK INHIBITORS AND THEIR USE FOR TREATING PAIN AND INFLAMMATION OMEROS MEDICAL SYSTEMS, INC. (US) 2000-04-27 WO claimed
EP-0889887-A1 NOVEL TREATMENT FOR CNS INJURIES SMITHKLINE BEECHAM CORPORATION (US) 1999-01-13 EP claimed
WO-1997035855-A1 NOVEL TREATMENT FOR CNS INJURIES SMITHKLINE BEECHAM CORPORATION (US) 1997-10-02 WO claimed
US-5656644-A CYTOKINE SUPPRESSORS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-12 US claimed
EP-0623126-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS CYTOKINE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-11-09 EP claimed
WO-1993014081-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS CYTOKINE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-07-22 WO claimed