SCHEMBL9521112

SCHEMBL9521112

CCOC(=O)COC[C@@H]1C[C@@H](O[Si](C)(C)C(C)(C)C)CN1C(=O)OCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.38
POLB P06746 1/20 0.38
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37
PDK3 Q15120 1/20 0.37
PDK4 Q16654 1/20 0.37
ITGB1 P05556 6/20 0.36
ITGA5 P08648 6/20 0.36
ITGB3 P05106 5/20 0.36
ITGAV P06756 5/20 0.36
ITGB5 P18084 3/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
TSHR P16473 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
USP2 O75604 1/20 0.35
ITGA2B P08514 2/20 0.35
AGTR2 P50052 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14348092 0.86 ABCB1 (0.42) ABCB1POLBPDK1PDK2PDK3
SCHEMBL9639974 0.85 ABCB1 (0.41) ABCB1POLBPDK1PDK2PDK3
SCHEMBL18962 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL15958482 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL9370028 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL9026282 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL8833139 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL9370027 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL29254 0.84 ABCB1 (0.43) ABCB1POLBPDK1PDK2PDK3
SCHEMBL9369164 0.83 ABCB1 (0.40) ABCB1POLBPDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272456-B1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid compounds and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-03-31 EP disclosed
US-4822787-A 3-pyrrolidinylthio-1-azabicyclo(3.2.0)-hept-2-ene-2-carboxylic acid compounds and antimicrobial activity thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-04-18 US disclosed
EP-0272456-A1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid compounds and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1988-06-29 EP disclosed