SCHEMBL9521783

SCHEMBL9521783

Cc1ccc(-c2nc(CCC(=O)c3ccc(C=O)cc3)c(C)o2)o1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.36
KDM4E B2RXH2 6/20 0.36
GAA P10253 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
PPARG P37231 6/20 0.33
PPARA Q07869 5/20 0.33
PPARD Q03181 2/20 0.32
KAT8 Q9H7Z6 1/20 0.32
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523037 0.83 PPARG (0.46) ALDH1A1KDM4ELMNAMAPTPPARG
SCHEMBL5795341 0.83 KDM4E (0.54) KDM4EPPARGPPARAPPARDFFAR1
SCHEMBL9520639 0.82 PIM1 (0.43) RAB9A
SCHEMBL9520645 0.82 PIM1 (0.43) RAB9A
SCHEMBL10480772 0.82 KDM4E (0.53) KDM4EPPARGPPARAPPARDFFAR1
SCHEMBL10480771 0.81 KDM4E (0.52) KDM4EPPARGPPARAPPARDFFAR1
SCHEMBL9521218 0.78 PPARA (0.49) MAPTPPARGPPARAPPARD
SCHEMBL9520936 0.78 PPARG (0.43) ALDH1A1KDM4EMAPTPPARGPPARA
SCHEMBL9523122 0.75 PPARG (0.44) ALDH1A1MAPTPPARGPPARAFFAR1
SCHEMBL9787633 0.74 HDAC1 (0.44) ALDH1A1KDM4EGAALMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0332332-B1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1993-03-31 EP disclosed
US-5130379-A Anticholesterol agents and antidiabetic agents PFIZER INC. (US) 1992-07-14 US disclosed
US-5036079-A Anticholesterol PFIZER INC. (US) 1991-07-30 US disclosed
WO-1991003474-A1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1991-03-21 WO disclosed