Oxalic Acid

Oxalic Acid

SCHEMBL9524892

Clc1cccc(C(c2ccc3nnn(OCc4ccccc4)c3c2)n2ccnc2)c1.Clc1cccc(C(c2ccc3nnn(OCc4ccccc4)c3c2)n2ccnc2)c1.O=C(O)C(=O)O.O=C(O)C(=O)O.O=C(O)C(=O)O

nearest known ligand 0.47

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Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.47
CYP3A4 P08684 2/20 0.47
CYP26A1 O43174 2/20 0.47
CYP2C8 P10632 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP24A1 Q07973 1/20 0.47
CYP26B1 Q9NR63 1/20 0.47
ACE P12821 1/20 0.45
EMG1 Q92979 1/20 0.45
CNR1 P21554 3/20 0.44
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 2/20 0.38
CYP17A1 P05093 2/20 0.38
NR1I2 O75469 1/20 0.38
USP2 O75604 1/20 0.38
ABCB11 O95342 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9524883 1.00 CYP19A1 (0.47) CYP19A1CYP3A4CYP26A1CYP2C8CYP2D6
SCHEMBL9523819 0.81 CYP19A1 (0.50) CYP19A1CYP3A4CYP26A1CYP2C8CYP2D6
SCHEMBL9527065 0.80 CYP17A1 (0.48) CYP3A4CYP26A1KMT2ASMN1; SMN2CYP17A1
SCHEMBL9524756 0.79 CYP19A1 (0.60) CYP19A1CYP3A4CYP26A1CYP2C8CYP2D6
Oxalic Acid SCHEMBL27275153 0.74 CYP19A1 (0.51) CYP19A1CYP3A4CYP26A1CNR1KMT2A
Oxalic Acid SCHEMBL9527036 0.74 CYP19A1 (0.51) CYP19A1CYP3A4CYP26A1CNR1KMT2A
SCHEMBL14092717 0.73 CYP19A1 (0.59) CYP19A1CYP3A4CYP26A1CYP2C8CYP2D6
SCHEMBL3279238 0.72 CYP19A1 (0.60) CYP19A1CYP3A4CYP26A1CYP2C8CYP2D6
Oxalic Acid SCHEMBL9868434 0.71 CYP19A1 (0.48) CYP19A1CYP3A4CYP26A1CNR1KMT2A
Oxalic Acid SCHEMBL27268074 0.71 CYP19A1 (0.48) CYP19A1CYP3A4CYP26A1CNR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293978-B1 (1H-AZOL-1-YLMETHYL)SUBSTITUTED BENZOTRIAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-09-15 EP disclosed
US-5039677-A Estrogen inhibitor JANSSEN PHARMACEUTICA N.V. (CA) 1991-08-13 US disclosed
US-4943574-A AROMATASE INHIBITORS, ESTROGEN DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-24 US disclosed
EP-0293978-A2 (1H-azol-1-ylmethyl)substituted benzotriazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-12-07 EP disclosed