SCHEMBL9525291

SCHEMBL9525291

CCCCCCc1ccc(NC(=O)OCCNC(=O)OCCN(C(=O)c2cncc(Br)c2)c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
POLB P06746 1/20 0.43
CHRNA7 P36544 2/20 0.40
ALDH1A1 P00352 1/20 0.40
ADRB2 P07550 1/20 0.40
CASP3 P42574 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TRPV1 Q8NER1 5/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
S1PR1 P21453 1/20 0.38
RECQL P46063 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
CFTR P13569 1/20 0.37
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525133 0.91 NPC1 (0.47) TSHRNPC1RAB9AMAPT
SCHEMBL9525766 0.88 POLB (0.54) POLBALDH1A1CASP3NPC1RAB9A
SCHEMBL9528113 0.86 NPC1 (0.43) TSHRPOLBALDH1A1NPC1RAB9A
Hydrochloric Acid SCHEMBL9525055 0.85 TSHR (0.41) TSHRCHRNA7ALDH1A1ADRB2NPC1
SCHEMBL9525835 0.83 HRH3 (0.42) POLBALDH1A1ADRB2NPC1RAB9A
SCHEMBL9525171 0.82 NPC1 (0.41) POLBALDH1A1ADRB2NPC1RAB9A
SCHEMBL9525526 0.80 POLB (0.44) POLBALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL9525476 0.80 POLB (0.46) TSHRPOLBALDH1A1CASP3NPC1
SCHEMBL9525705 0.80 NPC1 (0.47) TSHRPOLBALDH1A1CASP3NPC1
SCHEMBL9525183 0.79 POLB (0.45) TSHRPOLBALDH1A1CASP3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed