SCHEMBL9525869

SCHEMBL9525869

O=C(OCCN(C(=O)c1cncc(Br)c1)c1ccccc1)N(CCO)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.44
ALOX15 P16050 1/20 0.44
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.40
POLB P06746 3/20 0.40
HCAR2 Q8TDS4 1/20 0.40
KMT2A Q03164 2/20 0.39
TSHR P16473 3/20 0.39
GAA P10253 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
EGFR P00533 1/20 0.38
MEN1 O00255 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525204 0.92 KMT2A (0.45) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9525897 0.89 GAA (0.43) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9526168 0.86 HTT (0.46) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9525194 0.85 HTT (0.45) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9525705 0.85 NPC1 (0.47) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9524303 0.83 HTT (0.50) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9525476 0.83 POLB (0.46) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9528250 0.83 KDR (0.41) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9525183 0.83 POLB (0.45) HTTALOX15NPC1RAB9ASMN1; SMN2
SCHEMBL9524110 0.82 NPC1 (0.46) HTTALOX15NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed