SCHEMBL9526323

SCHEMBL9526323

COc1c(C)cnc(CSc2nc3cc(OC(F)F)c(OC(F)F)cc3[nH]2)c1C

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 3/20 0.66
ATP4A P20648 8/20 0.49
ATP4B P51164 8/20 0.49
ATP1A1 P05023 6/20 0.49
ATP1B1 P05026 6/20 0.49
ATP1A3 P13637 6/20 0.49
ATP1B2 P14415 6/20 0.49
ATP1A2 P50993 6/20 0.49
ATP1B3 P54709 6/20 0.49
FXYD2 P54710 6/20 0.49
ATP1A4 Q13733 6/20 0.49
CYP2C9 P11712 6/20 0.40
CYP1A2 P05177 5/20 0.40
CYP3A4 P08684 5/20 0.40
CYP2C19 P33261 5/20 0.40
WDR5 P61964 3/20 0.40
KMT2A Q03164 3/20 0.40
HTT P42858 2/20 0.40
KDM4E B2RXH2 1/20 0.40
DDAH1 O94760 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527971 0.98 BRS3 (0.63) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL6882572 0.93 BRS3 (0.56) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL6882415 0.92 BRS3 (0.55) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL27697403 0.91 BRS3 (0.54) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL6882809 0.91 BRS3 (0.54) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL6881008 0.91 BRS3 (0.54) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL9528548 0.87 BRS3 (0.62) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL9527121 0.86 BRS3 (0.69) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL9527490 0.86 BRS3 (0.60) BRS3ATP4AATP4BATP1A1ATP1B1
SCHEMBL10502388 0.85 BRS3 (0.52) BRS3ATP4AATP4BATP1A1ATP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0134400-B1 FLUOROALKOXYSUBSTITUTED PYRIDYLMETHYLTHIO-(OR SULFINYL-)BENZIMIDAZOLES HAVING A SECRETOLYTIC ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1993-03-24 EP disclosed
US-4555518-A ANTIULCER AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1985-11-26 US disclosed
EP-0134400-A2 Fluoroalkoxysubstituted pyridylmethylthio-(or sulfinyl-)benzimidazoles having a secretolytic activity Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1985-03-20 EP disclosed